Agents
Non-Selective α-Adrenergic Receptor Antagonists
- Phenoxybenzamine (see Phenoxybenzamine, [[Phenoxybenzamine]])
- Phentolamine (Regitine) (see Phentolamine, [[Phentolamine]])
- Tolazoline
- Trazodone (see Trazodone, [[Trazodone]])
- Typical and Atypical Antipsychotics
- Olanzapine (Zyprexa) (see Olanzapine, [[Olanzapine]])
- Potent Serotonin 5-HT2A and 5-HT2C, Dopamine D1-4, Histamine H1, and α1-Adrenergic Receptor Antagonism
- Moderate Serotonin 5-HT3 and Muscarinic M1-5 Receptor Antagonism
- Weak Binding to GABA-A, BZD, and β-Adrenergic Receptors
- Quetiapine (Seroquel) (see Quetiapine, [[Quetiapine]])
- Brain Serotonin 5-HT1A and 5-HT2, Dopamine D1 and D2, Histamine H1, and α1 and α2 Adrenergic Receptor Antagonism
- Risperidone (Risperdal) (see Risperidone, [[Risperidone]])
- Potent Serotonin 5-HT2, Dopamine D2, Adrenergic α1/α2, Histamine Receptor Antagonism
- Low-Moderate Serotonin 5-HT1C/5-HT1D/5-HT1A Receptor Antagonism
- Weak Dopamine D1 Receptor Antagonism
- Olanzapine (Zyprexa) (see Olanzapine, [[Olanzapine]])
Selective α1-Adrenergic Receptor Antagonists (see α1-Adrenergic Receptor Antagonists, [[α1-Adrenergic Receptor Antagonists]])
- Alfuzosin (Uroxatral) (see Alfuzosin, [[Alfuzosin]])
- Doxazosin (Cardura) (see Doxazosin, [[Doxazosin]])
- Prazosin (Minipress, Vasoflex, Pressin, Hypovase) (see Prazosin, [[Prazosin]])
- Silodosin (Rapaflo) (see Silodosin, [[Silodosin]])
- Tamsulosin (Flomax) (see Tamsulosin, [[Tamsulosin]])
- Terazosin (Hytrin) (see Terazosin, [[Terazosin]])
Selective α2-Adrenergic Receptor Antagonists
- Atipamezole (Antisedan)
- Idazoxan
- Mirtazapine (Remeron) (see Mirtazapine, [[Mirtazapine]])
- Yohimbine (Actibine, Erex, Testomar, Yocon, Yohimar, Yohimbe) (see Yohimbine, [[Yohimbine]])

References
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